IEM 1754 2HBr

CAS No. 162831-31-4

IEM 1754 2HBr( IEM-1754 dihydrobromide | IEM 1754 dihydrobromide )

Catalog No. M17347 CAS No. 162831-31-4

IEM 1754 2HBr is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 29 Get Quote
5MG 43 Get Quote
10MG 67 Get Quote
25MG 147 Get Quote
50MG 239 Get Quote
100MG 356 Get Quote
500MG 1053 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    IEM 1754 2HBr
  • Note
    Research use only, not for human use.
  • Brief Description
    IEM 1754 2HBr is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.
  • Description
    IEM-1754 2HBr is a voltage-dependent open-channel blocker of AMPA receptors. It acts by selectively blocking GluR2 subunit-lacking (Ca2+-permeable) receptors.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    IEM-1754 dihydrobromide | IEM 1754 dihydrobromide
  • Pathway
    GPCR/G Protein
  • Target
    Antibacterial
  • Recptor
    mGluR1| mGluR3
  • Research Area
    Others-Field
  • Indication
    ——

Chemical Information

  • CAS Number
    162831-31-4
  • Formula Weight
    412.25
  • Molecular Formula
    C16H30N2·2HBr
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (242.57 mM)
  • SMILES
    Br.Br.NCCCCCNCC12CC3CC(CC(C3)C1)C2
  • Chemical Name
    N-(Tricyclo[3.3.1.13,7]dec-1-ylmethyl)-1,5-pentanediamine dihydrobromide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Magazanik LG, et al. J Physiol, 1997, 505( Pt 3), 655-663.
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